SCHEMBL29800024

SCHEMBL29800024

CON(C)C(=O)c1cccc(CNc2ncnc(N)c2-c2ccc(Oc3ccccc3)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.49
EGFR P00533 5/20 0.47
KCNH2 Q12809 3/20 0.47
TEC P42680 1/20 0.46
BMX P51813 1/20 0.46
CD69 Q07108 1/20 0.46
ITK Q08881 1/20 0.46
ERBB4 Q15303 1/20 0.46
GP6 Q9HCN6 1/20 0.46
NUDT5 Q9UKK9 1/20 0.46
AURKA O14965 1/20 0.42
RPS6KB1 P23443 1/20 0.42
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14165581 1.00 BTK (0.49) BTKEGFRKCNH2TECBMX
SCHEMBL14165742 0.88 BTK (0.53) BTKEGFRKCNH2TECBMX
SCHEMBL14165706 0.87 BTK (0.53) BTKEGFRKCNH2TECBMX
SCHEMBL14241647 0.85 BTK (0.62) BTKEGFRKCNH2TECBMX
SCHEMBL14165903 0.83 BTK (0.51) BTKEGFRKCNH2TECBMX
SCHEMBL14165423 0.83 BTK (0.50) BTKEGFRKCNH2TECBMX
SCHEMBL14165422 0.83 BTK (0.50) BTKEGFRKCNH2TECBMX
SCHEMBL14241716 0.83 BTK (0.57) BTKEGFRKCNH2TECBMX
SCHEMBL24363478 0.82 BTK (0.50) BTKEGFRKCNH2TECBMX
SCHEMBL28156821 0.78 BTK (0.52) BTKEGFRKCNH2TECBMX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4056562-A1 HETEROCYCLIC INHIBITORS OF BRUTON'S TYROSINE KINASE Merck Patent GmbH (DE) 2022-09-14 EP disclosed