SCHEMBL29800784

SCHEMBL29800784

COc1ccc2c(c1)Oc1cc(F)ccc1N=C2N1CCN(CC(C)(C)C(=O)O)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 15/20 1.00
HRH1 P35367 10/20 0.81
HTR2C P28335 6/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23242585 1.00 HTR2A (1.00) HTR2AHRH1HTR2C
SCHEMBL10194141 0.94 HTR2A (0.89) HTR2AHRH1HTR2C
SCHEMBL10194091 0.93 HTR2A (0.87) HTR2AHRH1HTR2C
SCHEMBL23242581 0.93 HTR2A (1.00) HTR2AHRH1HTR2C
SCHEMBL23242617 0.92 HTR2A (0.86) HTR2AHRH1HTR2C
SCHEMBL29800676 0.92 HTR2A (0.86) HTR2AHRH1HTR2C
SCHEMBL23242609 0.90 HTR2A (1.00) HTR2AHRH1HTR2C
SCHEMBL29800763 0.90 HTR2A (1.00) HTR2AHRH1HTR2C
SCHEMBL10194105 0.89 HTR2A (0.81) HTR2AHRH1HTR2C
SCHEMBL23242501 0.89 HTR2A (1.00) HTR2AHRH1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114929688-B 3- (4- (11H-dibenzo [ b, e ] [1,4] azepin-6-yl) piperazin-1-yl) -and 3- (4- (dibenzo [ b, f ] [1,4] oxazepin/thiazepin/diazepin-11-yl) piperazin-1-yl) -propionic acid derivatives as H1 and 5-HT 2A-receptor modulators for the treatment of sleep disorders 阿莱瑞恩公司 2024-11-01 CN disclosed
CN-114929688-A 3- (4- (11H-dibenzo [ b, e ] [1,4] azepin-6-yl) piperazin-1-yl) -and 3- (4- (dibenzo [ b, f ] [1,4] oxazepin/thiazepin/diazepin-11-yl) piperazin-1-yl) -propionic acid derivatives as H1 and 5-HT 2A-receptor modulators for the treatment of sleep disorders 阿莱瑞恩公司 2022-08-19 CN disclosed