SCHEMBL29802986

SCHEMBL29802986

COc1ccc(/C=C/C(=O)c2cccc(O)c2)c(OC)c1OC

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 2/20 0.71
NR1H4 Q96RI1 2/20 0.70
CHRNA7 P36544 3/20 0.65
CYP1A1 P04798 2/20 0.65
CYP1A2 P05177 2/20 0.65
CYP2D6 P10635 2/20 0.65
CYP1B1 Q16678 2/20 0.65
CYP3A4 P08684 1/20 0.65
DPP4 P27487 1/20 0.63
MAOB P27338 1/20 0.59
LMNA P02545 2/20 0.58
NPC1 O15118 1/20 0.58
TP53 P04637 1/20 0.58
RAB9A P51151 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
ALDH1A1 P00352 1/20 0.58
NTSR1 P30989 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
RELA Q04206 1/20 0.58
ABCB1 P08183 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21643397 1.00 ABCG2 (0.71) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL21643325 0.91 NR1H4 (0.62) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL29730952 0.91 NR1H4 (0.62) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL29803485 0.89 NR1H4 (0.66) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL21643422 0.89 NR1H4 (0.66) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL7097693 0.86 ABCG2 (0.69) ABCG2NR1H4CHRNA7CYP1A1CYP1A2
SCHEMBL21643256 0.86 ABCG2 (0.70) ABCG2NR1H4CYP1A2CYP3A4DPP4
SCHEMBL29803039 0.86 ABCG2 (0.70) ABCG2NR1H4CYP1A2CYP3A4DPP4
SCHEMBL1764954 0.85 ABCG2 (0.86) ABCG2CHRNA7CYP1A1CYP1A2CYP2D6
SCHEMBL28796418 0.85 ABCG2 (0.86) ABCG2CHRNA7CYP1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114746103-A Rapafucin derivative compounds and methods of use thereof 约翰霍普金斯大学 2022-07-12 CN disclosed