SCHEMBL2980467

SCHEMBL2980467

COc1ccc(-c2cncc(C#N)c2Nc2ccc3[nH]ccc3c2)cc1OCCN1CCN(C)CC1

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PRKCQ Q04759 20/20 0.79
PRKCD Q05655 10/20 0.79
PRKCH P24723 3/20 0.75
PRKCE Q02156 3/20 0.75
PRKCB P05771 2/20 0.58
LCK P06239 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2979910 0.95 PRKCQ (0.78) PRKCQPRKCDPRKCHPRKCEPRKCB
SCHEMBL2975252 0.94 PRKCQ (0.79) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2981587 0.93 PRKCQ (0.78) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2990473 0.93 PRKCQ (0.76) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2988008 0.93 PRKCQ (0.76) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2984296 0.92 PRKCQ (0.75) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2979959 0.88 PRKCQ (1.00) PRKCQPRKCDPRKCHPRKCEPRKCB
SCHEMBL2980190 0.88 PRKCQ (1.00) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2983277 0.87 PRKCQ (0.86) PRKCQPRKCDPRKCHPRKCE
SCHEMBL2983052 0.87 PRKCQ (0.79) PRKCQPRKCDPRKCHPRKCEPRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029543-B1 SUBSTITUTED 3-CYANOPYRIDINES AS PROTEIN KINASE INHIBITORS WYETH LLC (US) 2015-11-18 EP claimed
US-7781591-B2 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC (US) 2010-08-24 US claimed
US-20070287708-A1 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC 2007-12-13 US claimed
US-7781591-B2 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC (US) 2010-08-24 US disclosed
US-20070287708-A1 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC 2007-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070287708-A1 Substituted 3-cyanopyridines as protein kinase inhibitors CNKSR1, MAP3K1, MAP3K7 PRKCQ 165/4885PRKCD 323/4885PRKCH 64/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.