SCHEMBL298246

SCHEMBL298246

CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(F)c(C(F)(F)F)c4)cc23)c1F

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 12/20 0.79
BRAF P15056 2/20 0.79
RIPK2 O43353 1/20 0.79
ABCB11 O95342 1/20 0.79
EGFR P00533 1/20 0.79
KRAS P01116 1/20 0.79
RAF1 P04049 1/20 0.79
PGR P06401 1/20 0.79
RET P07949 1/20 0.79
CHRM2 P08172 1/20 0.79
ADORA3 P0DMS8 1/20 0.79
ARAF P10398 1/20 0.79
CHRM1 P11229 1/20 0.79
CHRM3 P20309 1/20 0.79
FECH P22830 1/20 0.79
KDR P35968 1/20 0.79
MAP2K2 P36507 1/20 0.79
TGFBR2 P37173 1/20 0.79
NEK2 P51955 1/20 0.79
MAP2K1 Q02750 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298389 0.94 BRAF (0.80) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL29898563 0.91 BRAF (0.83) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL298352 0.91 BRAF (0.83) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL20400626 0.91 CYP2C9 (0.86) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL10246457 0.90 CYP2C19 (0.84) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL298927 0.89 BRAF (0.89) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL21624540 0.89 CYP2C19 (0.76) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL21624513 0.89 CYP2C19 (0.73) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL29898574 0.89 CYP2C19 (0.76) CYP2C19BRAFRIPK2ABCB11EGFR
SCHEMBL30866607 0.89 CYP2C19 (0.73) CYP2C19BRAFRIPK2ABCB11EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed