SCHEMBL29831577

SCHEMBL29831577

Oc1nc(-c2cc(-c3ccon3)n(Cc3ccccc3F)n2)ncc1F

nearest known ligand 0.79

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GUCY1B2 O75343 20/20 0.79
GUCY1A2 P33402 20/20 0.79
GUCY1A1 Q02108 20/20 0.79
GUCY1B1 Q02153 20/20 0.79
OPRK1 P41145 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL250991 1.00 GUCY1B2 (0.79) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL15087556 0.92 GUCY1B2 (0.67) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL3439276 0.91 GUCY1B2 (0.72) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL3437255 0.91 GUCY1B2 (0.72) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL18405244 0.91 GUCY1B2 (0.72) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL10269507 0.91 GUCY1B2 (0.70) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL3437146 0.91 GUCY1B2 (0.70) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL15069463 0.90 GUCY1B2 (0.69) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL3436889 0.90 GUCY1B2 (0.69) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1
SCHEMBL17307870 0.89 GUCY1B2 (0.64) GUCY1B2GUCY1A2GUCY1A1GUCY1B1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118221665-A Methods and intermediates for preparing soluble guanylate cyclase stimulators 赛克里翁治疗有限公司 2024-06-21 CN disclosed
CN-118184645-A Methods and intermediates for preparing soluble guanylate cyclase stimulators 赛克里翁治疗有限公司 2024-06-14 CN disclosed
CN-111902410-B Methods and intermediates for preparing soluble guanylate cyclase stimulators 赛克里翁治疗有限公司 2024-04-19 CN disclosed
EP-3998260-B1 SGC STIMULATORS CYCLERION THERAPEUTICS INC (US) 2023-11-01 EP disclosed
CN-116942616-A Solid dispersion comprising sGC stimulators 赛克里翁治疗有限公司 2023-10-27 CN disclosed
CN-112105358-B Non-steroidal mineralocorticoid receptor antagonists alone or in combination for the treatment of muscle or neuromuscular diseases 拜耳公司 2023-10-13 CN disclosed
CN-116637077-A Solid dispersion comprising sGC stimulators 赛克里翁治疗有限公司 2023-08-25 CN disclosed
CN-116637076-A Solid dispersion comprising sGC stimulators 赛克里翁治疗有限公司 2023-08-25 CN disclosed
CN-109369635-B Compound or pharmaceutically acceptable salt thereof, application thereof and pharmaceutical composition 赛克里翁治疗有限公司 2023-06-30 CN disclosed
CN-109563086-B Process for preparing soluble guanylate cyclase stimulators 赛克里翁治疗有限公司 2023-05-23 CN disclosed
CN-109384778-B Use of a compound or a pharmaceutically acceptable salt thereof for the manufacture of a medicament for the treatment of a disease, health condition or disorder 赛克里翁治疗有限公司 2022-12-13 CN disclosed
CN-110016020-B Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 赛克里翁治疗有限公司 2022-07-26 CN disclosed