SCHEMBL29843962

SCHEMBL29843962

CC[C@@H](Nc1c(Nc2cccc(C(=O)N(C)C)c2O)c(=O)c1=O)c1cc(Br)co1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 20/20 1.00
CXCR2 P25025 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12262828 1.00 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12262801 1.00 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12262821 1.00 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12086644 0.90 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL31065211 0.89 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12263764 0.89 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12262822 0.89 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12262837 0.89 CXCR1 (1.00) CXCR1CXCR2
SCHEMBL12086725 0.89 CXCR2 (1.00) CXCR1CXCR2
SCHEMBL12262982 0.89 CXCR2 (0.79) CXCR1CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4686472-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR GRAFT-VERSUS-HOST DISEASE Dompé farmaceutici SpA (IT) 2026-02-04 EP claimed
EP-4646193-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID Dompé farmaceutici S.p.A. (IT) 2025-11-12 EP claimed
WO-2024146918-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID DOMPE' FARMACEUTICI SPA (IT) 2024-07-11 WO claimed
EP-4301351-A1 CXCL8 INHIBITOR AND PHARMACEUTICAL COMPOSITION THEREOF FOR USE IN THE TREATMENT OF SEIZURES Dompe' Farmaceutici SpA (IT) 2024-01-10 EP claimed
WO-2022184841-A1 CXCL8 INHIBITOR AND PHARMACEUTICAL COMPOSITION THEREOF FOR USE IN THE TREATMENT OF SEIZURES DOMPE' FARMACEUTICI SPA (IT) 2022-09-09 WO claimed
EP-4646193-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID Dompé farmaceutici S.p.A. (IT) 2025-11-12 EP disclosed
EP-4563594-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF TUMORS WITH LOW STROMAL CAV1 LEVELS Dompe' Farmaceutici SpA (IT) 2025-06-04 EP disclosed
WO-2024146918-A1 CXCL8 INHIBITORS FOR USE IN THE TREATMENT OF OCULAR MUCOUS MEMBRANE PEMPHIGOID AND/OR ORAL MUCOUS MEMBRANE PEMPHIGOID DOMPE' FARMACEUTICI SPA (IT) 2024-07-11 WO disclosed
EP-4301351-A1 CXCL8 INHIBITOR AND PHARMACEUTICAL COMPOSITION THEREOF FOR USE IN THE TREATMENT OF SEIZURES Dompe' Farmaceutici SpA (IT) 2024-01-10 EP disclosed
WO-2022184841-A1 CXCL8 INHIBITOR AND PHARMACEUTICAL COMPOSITION THEREOF FOR USE IN THE TREATMENT OF SEIZURES DOMPE' FARMACEUTICI SPA (IT) 2022-09-09 WO disclosed