SCHEMBL29844458

SCHEMBL29844458

COc1ccc(Cl)c(Cl)c1[C@@H]1CCN[C@H](CO)C1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.47
HTR2A P28223 11/20 0.47
HTR2B P41595 8/20 0.47
ADRA1A P35348 2/20 0.35
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
HTR1E P28566 1/20 0.33
HTR7 P34969 1/20 0.33
HTR3A P46098 1/20 0.33
HTR5A P47898 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217069 1.00 HTR2C (0.47) HTR2CHTR2AHTR2BADRA1ACHRNB4
SCHEMBL23217382 1.00 HTR2C (0.47) HTR2CHTR2AHTR2BADRA1ACHRNB4
SCHEMBL23216339 0.88 HTR2A (0.56) HTR2CHTR2AHTR2BADRA1AHTR1A
SCHEMBL29768478 0.88 HTR2A (0.56) HTR2CHTR2AHTR2BADRA1AHTR1A
SCHEMBL23227264 0.87 HTR2C (0.49) HTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL23217143 0.86 HTR2C (0.50) HTR2CHTR2AHTR2B
Hydrochloric Acid SCHEMBL29845008 0.86 HTR2C (0.50) HTR2CHTR2AHTR2B
SCHEMBL29768399 0.86 HTR2A (0.43) HTR2CHTR2AHTR2BADRA1ACHRNB4
SCHEMBL23216843 0.85 HTR2A (0.45) HTR2CHTR2AHTR2BADRA1ACHRNB4
SCHEMBL23216481 0.85 HTR2A (0.43) HTR2CHTR2AHTR2BADRA1ACHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4041405-A1 ARYL HETEROBICYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. Shaw Research, LLC (US) 2022-08-17 EP disclosed