SCHEMBL29847016

SCHEMBL29847016

C=CC(=O)Nc1cccc(-c2cccc3cnc(Nc4ccc(N5CCN(C)CC5)cc4)nc23)c1

nearest known ligand 0.85

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.85
FGFR2 P21802 3/20 0.82
FGFR1 P11362 3/20 0.80
KDR P35968 3/20 0.80
BTK Q06187 5/20 0.72
JAK2 O60674 3/20 0.69
BRD4 O60885 1/20 0.69
JAK3 P52333 5/20 0.65
JAK1 P23458 1/20 0.64
TYK2 P29597 1/20 0.64
BLK P51451 1/20 0.63
BMX P51813 1/20 0.63
FLT3 P36888 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16514922 1.00 EGFR (0.85) EGFRFGFR2FGFR1KDRBTK
Hydrochloric Acid SCHEMBL16513760 0.99 EGFR (0.84) EGFRFGFR2FGFR1KDRBTK
Hydrochloric Acid SCHEMBL29847904 0.99 EGFR (0.84) EGFRFGFR2FGFR1KDRBTK
Maleic Acid SCHEMBL29848267 0.96 EGFR (0.79) EGFRFGFR2FGFR1KDRBTK
Maleic Acid SCHEMBL22464670 0.96 EGFR (0.79) EGFRFGFR2FGFR1KDRBTK
Maleic Acid SCHEMBL16514642 0.96 EGFR (0.79) EGFRFGFR2FGFR1KDRBTK
Fumaric Acid SCHEMBL16514646 0.96 EGFR (0.79) EGFRFGFR2FGFR1KDRBTK
SCHEMBL16514042 0.93 EGFR (0.73) EGFRFGFR2FGFR1KDRBTK
SCHEMBL29847829 0.93 EGFR (0.73) EGFRFGFR2FGFR1KDRBTK
SCHEMBL29848454 0.92 FGFR1 (0.79) EGFRFGFR2FGFR1KDRBTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109851617-B Chemical entities, compositions, and methods 润新生物公司 2022-08-16 CN disclosed