SCHEMBL29848786

SCHEMBL29848786

CCCCc1cnc(S(C)(=O)=O)nc1-c1cc(OC)c(=O)n(C)c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.44
PDE4B Q07343 3/20 0.36
BRD9 Q9H8M2 6/20 0.36
TLR8 Q9NR97 1/20 0.35
CREBBP Q92793 1/20 0.35
BRD7 Q9NPI1 2/20 0.34
BRD2 P25440 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE10A Q9Y233 2/20 0.34
BPTF Q12830 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16651614 1.00 BRD4 (0.44) BRD4PDE4BBRD9TLR8CREBBP
SCHEMBL16651731 0.94 BRD4 (0.46) BRD4PDE4BBRD9CREBBPBRD7
SCHEMBL16651403 0.86 BRD4 (0.53) BRD4BRD9CREBBP
SCHEMBL29848844 0.86 BRD4 (0.53) BRD4BRD9CREBBP
SCHEMBL16650991 0.85 BRD4 (0.43) BRD4PDE4BPDE4APDE4CPDE4D
SCHEMBL29848752 0.85 BRD4 (0.43) BRD4PDE4BPDE4APDE4CPDE4D
SCHEMBL29848815 0.84 BRD4 (0.40) BRD4
SCHEMBL16651256 0.84 BRD4 (0.40) BRD4
SCHEMBL16651201 0.83 CREBBP (0.37) BRD4PDE4BCREBBPPDE4APDE4C
SCHEMBL29848696 0.83 CREBBP (0.37) BRD4PDE4BCREBBPPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240182490-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2024-06-06 US disclosed
US-11884680-B2 Bromodomain inhibitors CELGENE QUANTICEL RESEARCH, INC. (US) 2024-01-30 US disclosed
US-20220315601-A1 BROMODOMAIN INHIBITORS CELGENE QUANTICEL RESEARCH, INC. (US) 2022-10-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240182490-A1 BROMODOMAIN INHIBITORS BRD3, EP300, BRPF3 BRD4 5/4885PDE4B 2787/4885BRD9 19/4885
US-20220315601-A1 BROMODOMAIN INHIBITORS BRD3, EP300, BRPF3 BRD4 5/4885PDE4B 2787/4885BRD9 19/4885
US-11884680-B2 Bromodomain inhibitors BRD3, EP300, BRPF3 BRD4 5/4885PDE4B 2787/4885BRD9 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.