SCHEMBL29857789

SCHEMBL29857789

C[C@H](Oc1cc(Br)cnc1[N+](=O)[O-])c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.42
CGAS Q8N884 1/20 0.41
MAPT P10636 3/20 0.36
HTT P42858 3/20 0.34
LMNA P02545 1/20 0.34
CYP17A1 P05093 2/20 0.34
CYP19A1 P11511 2/20 0.34
CRHBP P24387 1/20 0.34
CRHR2 Q13324 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KMT2A Q03164 1/20 0.34
KCNA5 P22460 2/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
ESR2 Q92731 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26916894 1.00 LRRK2 (0.42) LRRK2CGASMAPTHTTLMNA
SCHEMBL29857938 1.00 LRRK2 (0.42) LRRK2CGASMAPTHTTLMNA
SCHEMBL26917000 1.00 LRRK2 (0.42) LRRK2CGASMAPTHTTLMNA
SCHEMBL26916891 1.00 LRRK2 (0.42) LRRK2CGASMAPTHTTLMNA
SCHEMBL26916901 0.88 LRRK2 (0.40) LRRK2MAPTHTTLMNAKMT2A
SCHEMBL26916906 0.88 LRRK2 (0.40) LRRK2MAPTHTTLMNAKMT2A
SCHEMBL29857833 0.87 LRRK2 (0.35) LRRK2MAPTHTTLMNAKMT2A
SCHEMBL26917105 0.87 LRRK2 (0.35) LRRK2MAPTHTTLMNAKMT2A
SCHEMBL29857862 0.87 LRRK2 (0.35) LRRK2MAPTHTTLMNAKMT2A
SCHEMBL26916824 0.87 LRRK2 (0.35) LRRK2MAPTHTTLMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4288437-A1 MAP4K1 INHIBITORS Bayer Aktiengesellschaft (DE) 2023-12-13 EP disclosed
WO-2022167627-A1 MAP4K1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2022-08-11 WO disclosed