SCHEMBL298623

SCHEMBL298623

O=C(O)c1ccnc2c(O)cccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 1.00
L3MBTL1 Q9Y468 4/20 1.00
KDM4A O75164 2/20 1.00
EGLN1 Q9GZT9 2/20 1.00
RAB9A P51151 1/20 1.00
HIF1AN Q9NWT6 1/20 1.00
KDM6B O15054 1/20 0.75
KDM6A O15550 1/20 0.75
TET3 O43151 1/20 0.75
KDM4B O94953 1/20 0.75
KDM5C P41229 1/20 0.75
KDM4D Q6B0I6 1/20 0.75
TET2 Q6N021 1/20 0.75
ALKBH5 Q6P6C2 1/20 0.75
TET1 Q8NFU7 1/20 0.75
FTO Q9C0B1 1/20 0.75
KDM4C Q9H3R0 1/20 0.75
KDM2A Q9Y2K7 1/20 0.75
KDM3A Q9Y4C1 1/20 0.75
PSMD14 O00487 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6068195 0.86 KDM4E (1.00) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL29349767 0.86 KDM4E (1.00) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL69905 0.85 KDM4E (0.74) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL11159839 0.84 KDM4E (1.00) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL8617622 0.83 KDM4E (0.71) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL23754362 0.81 KDM4E (0.68) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL7373143 0.81 KDM4E (0.68) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL5761539 0.81 KDM4E (0.68) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL15129840 0.81 KDM4E (0.68) KDM4EL3MBTL1KDM4AEGLN1RAB9A
SCHEMBL4519716 0.81 KDM4E (0.68) KDM4EL3MBTL1KDM4AEGLN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 42 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114534694-B Hydroxyquinoline filler and preparation method and application thereof 万华化学集团股份有限公司 2024-08-16 CN claimed
CN-117567994-A Low-conductivity antifreezing cooling liquid and preparation method thereof 道骐科技有限公司 2024-02-20 CN claimed
CN-114534694-A Hydroxyquinoline filler and preparation method and application thereof 万华化学集团股份有限公司 2022-05-27 CN claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
US-3956420-A CPOLYOLEFIN COMPOSITION FOR ELECTRICAL INSULATIONFERROCENE, 8-SUBSTITUTED QUINOLINE DAINICHI-NIPPON CABLES, LTD. (JA) 1976-05-11 US claimed
CN-114534694-B Hydroxyquinoline filler and preparation method and application thereof 万华化学集团股份有限公司 2024-08-16 CN disclosed
CN-117567994-A Low-conductivity antifreezing cooling liquid and preparation method thereof 道骐科技有限公司 2024-02-20 CN disclosed
WO-2023247488-A1 N-(2-(3-CYANO-2-AZABICYCLO[3.1.0]HEXAN-2-YL)-2-OXOETHYL)- QUINOLINE-4-CARBOXAMIDES ASTRAZENECA AB (SE) 2023-12-28 WO disclosed
WO-2023002045-A1 FIBROBLAST ACTIVATION PROTEIN INHIBITORS AND USE THEREOF 3B PHARMACEUTICALS GMBH (DE) 2023-01-26 WO disclosed
EP-4122499-A1 FIBROBLAST ACTIVATION PROTEIN INHIBITORS AND USE THEREOF 3B Pharmaceuticals GmbH (DE) 2023-01-25 EP disclosed
CN-114534694-A Hydroxyquinoline filler and preparation method and application thereof 万华化学集团股份有限公司 2022-05-27 CN disclosed
EP-3230281-B1 1,3-THIAZOL-2-YL SUBSTITUTED BENZAMIDES BAYER AG (DE) 2021-05-26 EP disclosed
CN-1829712-A Nicotinamide derivatives useful as PDE4 inhibitors PFIZER (US) 2006-09-06 CN disclosed
US-20060178408-A1 Nicotinamide derivatives useful as pde4 inhibitors BARBER CHRISTOPHER G 2006-08-10 US disclosed
EP-1651640-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS Pfizer Limited (GB) 2006-05-03 EP disclosed
US-20050043326-A1 Compounds PFIZER INC 2005-02-24 US disclosed
WO-2005009994-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed
EP-1091958-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2001-04-18 EP disclosed
WO-2000001692-A1 SALTS OF PAROXETINE SMITHKLINE BEECHAM PLC (GB) 2000-01-13 WO disclosed
US-3956420-A CPOLYOLEFIN COMPOSITION FOR ELECTRICAL INSULATIONFERROCENE, 8-SUBSTITUTED QUINOLINE DAINICHI-NIPPON CABLES, LTD. (JA) 1976-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178408-A1 Nicotinamide derivatives useful as pde4 inhibitors PDE4A, PDE4B, PDE4C KDM4E 1010/4885L3MBTL1 4649/4885KDM4A 506/4885
US-20050043326-A1 Compounds NQO1, NAMPT, NNT KDM4E 3109/4885L3MBTL1 4529/4885KDM4A 3402/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.