SCHEMBL29862869

SCHEMBL29862869

COc1nc(Br)cnc1C=O

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 16/20 0.42
CCR5 P51681 1/20 0.39
EDNRA P25101 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21274185 1.00 CCR4 (0.42) CCR4CCR5EDNRA
SCHEMBL23213755 0.85 CCR4 (0.39) CCR4CCR5EDNRA
SCHEMBL29955754 0.83 POLB (0.37)
SCHEMBL6057013 0.83 POLB (0.37)
SCHEMBL23623967 0.81 CCR4 (0.39) CCR4CCR5EDNRA
SCHEMBL29952590 0.81 KCNJ1 (0.38) CCR4EDNRA
SCHEMBL1474575 0.81 KCNJ1 (0.38) CCR4EDNRA
SCHEMBL1474943 0.78 CCR4 (0.42) CCR4EDNRA
SCHEMBL21274427 0.78 KCNJ1 (0.33)
SCHEMBL29952408 0.78 CCR4 (0.42) CCR4EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024175043-A1 PYRIDOPYRIMIDINE DERIVATIVE AND USE THEREOF 广东东阳光药业股份有限公司 2024-08-29 WO disclosed
EP-4045037-A1 HETEROARYL-BIPHENYL AMINES FOR THE TREATMENT OF PD-L1 DISEASES ChemoCentryx, Inc. (US) 2022-08-24 EP disclosed