SCHEMBL29868077

SCHEMBL29868077

N[C@H](Cc1ccc(Cl)cc1Cl)C(=O)N1CC(c2ccccn2)C1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 13/20 0.61
HDAC1 Q13547 3/20 0.61
HDAC3 O15379 1/20 0.61
HDAC2 Q92769 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
AKT1 P31749 1/20 0.53
AKT2 P31751 1/20 0.53
AKT3 Q9Y243 1/20 0.53
MC4R P32245 2/20 0.48
DPP4 P27487 1/20 0.48
SPR P35270 1/20 0.47
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29868239 0.84 HDAC8 (0.67) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL4774443 0.79 HDAC8 (0.61) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL29868117 0.79 MC4R (0.58) MC4R
SCHEMBL29868385 0.78 HDAC8 (0.59) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL29868386 0.78 HDAC8 (0.59) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL29868228 0.78 HDAC8 (0.65) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL4778422 0.78 HDAC8 (0.59) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL4902706 0.77 HDAC8 (0.56) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL4795360 0.77 HDAC8 (0.56) HDAC8HDAC1HDAC3HDAC2HDAC6
SCHEMBL4779058 0.76 HDAC8 (1.00) HDAC8HDAC1HDAC3HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022178544-A1 NOVEL HETEROCYCLIC COMPOUNDS AND RELATED METHODS OF MANUFACTURE AND USE IN HDAC INHIBITION KLOTHO THERAPEUTICS, INC. (US) 2022-08-25 WO disclosed