SCHEMBL29883545

SCHEMBL29883545

O=C(C=Cc1cccc(-c2cnc3[nH]ccc3c2)c1)Nc1ccc(F)c(F)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 17/20 0.72
BTK Q06187 3/20 0.52
ITK Q08881 3/20 0.52
CDK7 P50613 2/20 0.52
PLK4 O00444 1/20 0.52
DCLK1 O15075 1/20 0.52
ROCK2 O75116 1/20 0.52
PRKD3 O94806 1/20 0.52
MAP4K4 O95819 1/20 0.52
PAK4 O96013 1/20 0.52
CHEK2 O96017 1/20 0.52
INSR P06213 1/20 0.52
CDK1 P06493 1/20 0.52
FES P07332 1/20 0.52
ROS1 P08922 1/20 0.52
PDGFRB P09619 1/20 0.52
PDGFRA P16234 1/20 0.52
FER P16591 1/20 0.52
CDK2 P24941 1/20 0.52
MARK3 P27448 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28882074 1.00 CDK8 (0.72) CDK8BTKITKCDK7PLK4
SCHEMBL28882043 0.92 CDK8 (0.79) CDK8BTKITKCDK7PLK4
SCHEMBL29883553 0.92 CDK8 (0.79) CDK8BTKITKCDK7PLK4
SCHEMBL28882008 0.90 CDK8 (0.71) CDK8BTKITKCDK7PLK4
SCHEMBL29883584 0.90 CDK8 (0.71) CDK8BTKITKCDK7PLK4
SCHEMBL28882270 0.90 CDK8 (0.71) CDK8BTKITKCDK7PLK4
SCHEMBL29883357 0.90 CDK8 (0.71) CDK8BTKITKCDK7PLK4
SCHEMBL28882039 0.90 CDK8 (0.82) CDK8BTKITKCDK7PLK4
SCHEMBL29883753 0.90 CDK8 (0.82) CDK8BTKITKCDK7PLK4
SCHEMBL29883352 0.88 CDK8 (0.69) CDK8BTKITKCDK7PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141197-B 3-aromatic heterocycle substituted phenyl derivative and preparation method and application thereof 安徽医科大学 2024-03-26 CN disclosed
CN-115141197-A 3-aromatic heterocyclic substituted phenyl derivative and preparation method and application thereof 安徽医科大学 2022-10-04 CN disclosed