SCHEMBL29888396

SCHEMBL29888396

O=c1[nH]cnc2c(F)c(-c3ccccc3F)c(Cl)cc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.50
PIM1 P11309 2/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
PAK4 O96013 1/20 0.47
ABL1 P00519 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
IGF1R P08069 1/20 0.47
MET P08581 1/20 0.47
PDGFRB P09619 1/20 0.47
FGFR1 P11362 1/20 0.47
PDGFRA P16234 1/20 0.47
PRKACA P17612 1/20 0.47
FLT1 P17948 1/20 0.47
LTK P29376 1/20 0.47
GRK5 P34947 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23415332 1.00 PARP1 (0.50) PARP1PIM1AURKADAPK3JAK2
SCHEMBL18395037 0.79 PARP1 (0.47) PARP1PIM1AURKADAPK3JAK2
SCHEMBL29888467 0.76 KRAS (0.39) MAP4K4SMN1; SMN2ALDH1A1KDM4E
SCHEMBL23464717 0.76 KRAS (0.39) MAP4K4SMN1; SMN2ALDH1A1KDM4E
SCHEMBL23465081 0.74 MAP4K4 (0.49) MAP4K4
SCHEMBL25779676 0.74 SMN1; SMN2 (0.40) MAP4K4SMN1; SMN2
SCHEMBL21415486 0.74 PARP1 (0.51) PARP1PIM1AURKADAPK3JAK2
SCHEMBL16637093 0.74 PARP1 (0.47) PARP1PIM1AURKADAPK3JAK2
SCHEMBL29810919 0.74 PARP1 (0.47) PARP1PIM1AURKADAPK3JAK2
SCHEMBL18128478 0.71 IP6K1 (0.56) PARP1PIM1AURKADAPK3JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114980976-A Covalent RAS inhibitors and uses thereof 锐新医药公司 2022-08-30 CN disclosed