SCHEMBL29889798

SCHEMBL29889798

O=C1CCOc2cc(OCc3ccccc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 17/20 1.00
GRM5 P41594 7/20 1.00
NPC1 O15118 1/20 1.00
ALDH1A1 P00352 1/20 1.00
HPGD P15428 1/20 1.00
NFKB1 P19838 1/20 1.00
RAB9A P51151 1/20 1.00
NFKB2 Q00653 1/20 1.00
RELA Q04206 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
MAOA P21397 3/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2326572 1.00 MAOB (1.00) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL22451525 0.92 MAOB (0.85) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL6836955 0.89 MAOB (0.81) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL30353218 0.89 MAOB (0.81) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL23905149 0.87 MAOB (0.77) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL23905167 0.87 MAOB (1.00) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL281588 0.86 MAOB (1.00) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL23906031 0.85 MAOB (0.74) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL23906233 0.84 MAOB (0.71) MAOBGRM5NPC1ALDH1A1HPGD
SCHEMBL16562137 0.82 MAOB (0.69) MAOBGRM5NPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115003295-B Novel chroman derivatives having estrogen receptor degrading activity and uses thereof 冰洲石生物科技公司 2025-05-06 CN disclosed
EP-4541795-A1 AROMATIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF IN PREPARATION OF ESTROGEN RECEPTOR DEGRADER Hinova Pharmaceuticals Inc. (CN) 2025-04-23 EP disclosed
WO-2024015409-A1 CHROMAN DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2024-01-18 WO disclosed
CN-117229286-A Aromatic compound, preparation method thereof and application thereof in preparation of estrogen receptor degradation agent 海创药业股份有限公司 2023-12-15 CN disclosed
CN-110770211-B Alpha, beta unsaturated amide compound 协和麒麟株式会社 2023-09-19 CN disclosed
CN-111039916-B Tricyclic spiro compounds 小野药品工业株式会社 2023-04-28 CN disclosed
EP-4126835-A1 INHIBITORS OF ANTIGEN PRESENTATION BY HLA-DR Janssen Pharmaceutica NV (BE) 2023-02-08 EP disclosed
CN-108430972-B Alpha, beta-unsaturated amide compound 协和麒麟株式会社 2022-12-27 CN disclosed
CN-115003295-A Novel chroman derivatives having estrogen receptor degrading activity and uses thereof 冰洲石生物科技公司 2022-09-02 CN disclosed