SCHEMBL29895473

SCHEMBL29895473

CC(C)(C)OC(=O)Nc1cccc(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.47
WDR77 Q9BQA1 1/20 0.47
AAK1 Q2M2I8 2/20 0.46
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
CA1 P00915 2/20 0.43
CA9 Q16790 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CA2 P00918 1/20 0.43
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
CYP17A1 P05093 1/20 0.42
SIRT2 Q8IXJ6 3/20 0.42
SIRT1 Q96EB6 2/20 0.42
CA12 O43570 1/20 0.42
NAMPT P43490 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1300326 1.00 PRMT5 (0.47) PRMT5WDR77AAK1HCRTR1HCRTR2
SCHEMBL27118089 0.87 PRMT5 (0.48) PRMT5WDR77AAK1CA1CA9
SCHEMBL30874514 0.87 CA1 (0.46) CA1CA9CA2CA12CYP3A4
SCHEMBL21318698 0.87 AAK1 (0.46) PRMT5WDR77AAK1HCRTR1HCRTR2
SCHEMBL3319977 0.86 PRMT5 (0.48) PRMT5WDR77AAK1CA1CA9
SCHEMBL595545 0.85 SIRT2 (0.47) PRMT5WDR77AAK1SIRT2CYP3A4
SCHEMBL12567525 0.85 AAK1 (0.48) PRMT5WDR77AAK1CA1CA9
SCHEMBL30561474 0.85 AAK1 (0.49) PRMT5WDR77AAK1HCRTR1HCRTR2
SCHEMBL21030001 0.85 AAK1 (0.49) PRMT5WDR77AAK1HCRTR1HCRTR2
SCHEMBL3321460 0.85 PRMT5 (0.46) PRMT5WDR77AAK1CA1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023043292-A1 PREPARATION METHOD FOR PYRIMIDINE-2-AMINE 기초과학연구원 2023-03-23 WO disclosed
CN-110506044-B BRD4 inhibitor and preparation and application thereof 中国科学院上海药物研究所 2022-07-05 CN disclosed