SCHEMBL29906555

SCHEMBL29906555

CCc1nc(N2CC3CC3C2)ccc1CC=O

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 2/20 0.34
KLKB1 P03952 13/20 0.34
HCRTR1 O43613 2/20 0.33
HCRTR2 O43614 2/20 0.33
PDE10A Q9Y233 1/20 0.32
RBP4 P02753 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23754018 1.00 SMPD3 (0.34) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL23768950 0.89 SMPD3 (0.39) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL26307974 0.83 SMPD3 (0.33) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL23754009 0.83 SMPD3 (0.33) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL29906648 0.83 SMPD3 (0.33) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL23754011 0.83 SMPD3 (0.33) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL23769540 0.83 KLKB1 (0.34) KLKB1
SCHEMBL23769616 0.82 SMPD3 (0.36) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL23754003 0.81 SMPD3 (0.36) SMPD3KLKB1HCRTR1HCRTR2PDE10A
SCHEMBL31357751 0.81 SMPD3 (0.36) SMPD3KLKB1HCRTR1HCRTR2PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116120287-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2025-01-28 CN disclosed
CN-116120287-A Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2023-05-16 CN disclosed
CN-115052873-A Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2022-09-13 CN disclosed