SCHEMBL29906606

SCHEMBL29906606

CCOC(=O)c1cn(Cc2ccc(N3CC4CC4C3)cc2C)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 8/20 0.46
NOTUM Q6P988 1/20 0.43
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
GABRA2 P47869 2/20 0.33
GABRB2 P47870 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23754033 1.00 KLKB1 (0.46) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL29906573 0.90 KLKB1 (0.45) KLKB1NOTUMKDM4EMAPTLMNA
SCHEMBL29906576 0.90 KLKB1 (0.45) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL23753982 0.90 KLKB1 (0.45) KLKB1NOTUMKDM4EMAPTLMNA
SCHEMBL23753990 0.90 KLKB1 (0.45) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL23754307 0.89 KLKB1 (0.44) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL29906616 0.89 KLKB1 (0.44) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL23754054 0.88 KLKB1 (0.60) KLKB1NOTUM
SCHEMBL23754073 0.88 KLKB1 (0.43) KLKB1NOTUMKDM4EMAPTALDH1A1
SCHEMBL26313088 0.88 KLKB1 (0.43) KLKB1NOTUMKDM4EMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116120287-B Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2025-01-28 CN disclosed
CN-116120287-A Heteroaromatic carboxamide derivatives as inhibitors of plasma kallikrein 勃林格殷格翰国际有限公司 2023-05-16 CN disclosed
EP-4103562-A1 HETEROAROMATIC CARBOXAMIDE DERIVATIVES AS PLASMA KALLIKREIN INHIBITORS Boehringer Ingelheim International GmbH (DE) 2022-12-21 EP disclosed
CN-115052873-A Heteroaromatic carboxamide derivatives as plasma kallikrein inhibitors 勃林格殷格翰国际有限公司 2022-09-13 CN disclosed