SCHEMBL29907107

SCHEMBL29907107

CNc1cc2c(nc1-c1cccc(C)c1C)c(-c1cnn(C)c1)nn2C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TYRO3 Q06418 9/20 0.36
AXL P30530 8/20 0.36
MERTK Q12866 6/20 0.36
PFKFB3 Q16875 1/20 0.34
HDAC8 Q9BY41 1/20 0.33
TTK P33981 3/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
MAP4K1 Q92918 1/20 0.32
GRM2 Q14416 1/20 0.32
NTRK1 P04629 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23211006 1.00 TYRO3 (0.36) TYRO3AXLMERTKPFKFB3HDAC8
SCHEMBL23210979 0.82 TYRO3 (0.39) TYRO3AXLMERTKPFKFB3
SCHEMBL29907078 0.82 TYRO3 (0.39) TYRO3AXLMERTKPFKFB3
SCHEMBL23249325 0.78 NTRK1 (0.32) TYRO3AXLMERTKNTRK1
SCHEMBL23210952 0.76 TYRO3 (0.40) TYRO3AXLMERTK
SCHEMBL29906967 0.76 MAP4K1 (0.49) AXLMAP4K1
SCHEMBL23210831 0.76 MAP4K1 (0.49) AXLMAP4K1
SCHEMBL23211013 0.72 KDM4E (0.40) TYRO3AXLMERTK
SCHEMBL30308766 0.69 MAPK1 (0.34)
SCHEMBL30308884 0.68 MAPK1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115835908-A Bicyclic heterocycles as FGFR inhibitors 因赛特公司 2023-03-21 CN disclosed
EP-4045151-A1 BICYCLIC HETEROCYCLES AS FGFR INHIBITORS Incyte Corporation (US) 2022-08-24 EP disclosed