SCHEMBL29907256

SCHEMBL29907256

OCCc1cccc2[nH]cnc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
DPP4 P27487 1/20 0.40
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
DRD4 P21917 3/20 0.38
DRD3 P35462 3/20 0.38
SLC40A1 Q9NP59 1/20 0.38
DRD2 P14416 2/20 0.38
PKM P14618 2/20 0.37
HTR1A P08908 2/20 0.37
BRD4 O60885 1/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856462 1.00 PARP1 (0.47) PARP1HTR2AHTR2CDPP4ADORA2A
SCHEMBL23124283 0.90 PARP1 (0.45) PARP1HTR2AHTR2CDPP4ADORA2A
SCHEMBL556764 0.87 PARP1 (0.51) PARP1HTR2AHTR2CDPP4ADORA2A
SCHEMBL3068250 0.82 PARP1 (0.47) PARP1HTR2AHTR2CDPP4ADORA2A
SCHEMBL7846859 0.80 PARP1 (0.50) PARP1HTR2AHTR2CADORA2AADORA1
SCHEMBL7856329 0.79 HTR2A (0.43) PARP1HTR2AHTR2CDRD4DRD3
SCHEMBL6043794 0.79 PARP1 (0.41) PARP1HTR2AHTR2CDPP4ADORA2A
SCHEMBL2820808 0.79 PARP1 (0.56) PARP1HTR2AHTR2CADORA2AADORA1
SCHEMBL31693421 0.78 HTR2A (0.47) PARP1HTR2AHTR2CADORA2ADRD3
SCHEMBL21941453 0.78 HTR2A (0.42) PARP1HTR2AHTR2CADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-120035595-A Thiazolo [5,4-d ] pyrimidine compounds, compositions comprising the same and uses thereof 蒙特利尔大学 2025-05-23 CN disclosed
EP-4326719-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE Université de Montréal (CA) 2024-02-28 EP disclosed
CN-117177973-A Pyrido [3,2-D ] pyrimidine compounds and their use for the treatment of proliferative disorders 蒙特利尔大学 2023-12-05 CN disclosed
WO-2022221939-A1 PYRIDO[3,2-D]PYRIMIDINE COMPOUNDS USES THEREOF FOR TREATING A PROLIFERATIVE DISEASE UNIVERSITE DE MONTREAL (CA) 2022-10-27 WO disclosed