SCHEMBL29907792

SCHEMBL29907792

COc1ccccc1CNC(=O)c1nc(Cl)c(-c2ccc(F)cc2)nc1N

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.66
ADORA1 P30542 3/20 0.66
ADORA2B P29275 1/20 0.66
ALDH1A1 P00352 4/20 0.49
HPGD P15428 3/20 0.49
KDM4E B2RXH2 2/20 0.49
HTT P42858 1/20 0.49
RCE1 Q9Y256 1/20 0.49
TP53 P04637 2/20 0.48
LMNA P02545 1/20 0.48
PLA2G1B P04054 1/20 0.48
ATG4B Q9Y4P1 1/20 0.48
MAPT P10636 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
POLB P06746 1/20 0.47
TSHR P16473 1/20 0.47
NPC1 O15118 2/20 0.47
GAA P10253 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MEN1 O00255 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22552058 1.00 ADORA2A (0.66) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL22551795 0.88 ADORA2A (0.59) ADORA2AADORA1ADORA2BHTTMAPT
SCHEMBL22551955 0.86 ADORA2A (0.83) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL29906692 0.86 ADORA2A (0.83) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL22552134 0.86 ADORA2A (0.74) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL29906736 0.86 ADORA2A (0.74) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL22552049 0.84 ADORA2A (0.76) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL21722355 0.83 ADORA2A (0.73) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL22551889 0.82 ADORA2A (0.61) ADORA2AADORA1ADORA2BALDH1A1HPGD
SCHEMBL21730176 0.82 ADORA2A (0.63) ADORA2AADORA1ADORA2BALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed