SCHEMBL29911990

SCHEMBL29911990

CN1CCN(c2cncc(-c3cccc(C(=O)Nc4cn(C)nc4-c4ccccn4)n3)c2)CC1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 19/20 0.53
KCNH2 Q12809 2/20 0.47
SCN9A Q15858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20085961 1.00 IRAK4 (0.53) IRAK4KCNH2SCN9A
SCHEMBL20085966 0.95 IRAK4 (0.53) IRAK4KCNH2
SCHEMBL29911962 0.95 IRAK4 (0.53) IRAK4KCNH2
SCHEMBL20085968 0.93 IRAK4 (0.56) IRAK4KCNH2SCN9A
SCHEMBL29912108 0.93 IRAK4 (0.56) IRAK4KCNH2SCN9A
SCHEMBL30261571 0.86 IRAK4 (0.58) IRAK4KCNH2
SCHEMBL20085939 0.86 IRAK4 (0.58) IRAK4KCNH2
SCHEMBL20085934 0.85 IRAK4 (0.57) IRAK4KCNH2
SCHEMBL20085954 0.85 IRAK4 (0.59) IRAK4KCNH2
SCHEMBL20086084 0.85 IRAK4 (0.54) IRAK4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115531387-A Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-12-30 CN disclosed
CN-110234637-B Pyrazole amide compounds useful as IRAK inhibitors 里格尔药品股份有限公司 2022-11-01 CN disclosed