SCHEMBL29919355

SCHEMBL29919355

C[Si](C)(C)CCOCn1c(=O)oc2cc(C[C@H](N)CN3C(=O)c4ccccc4C3=O)ccc21

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
USP2 O75604 1/20 0.37
HPGD P15428 1/20 0.37
MIF P14174 2/20 0.35
MAPT P10636 2/20 0.34
SIGMAR1 Q99720 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TNIK Q9UKE5 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
CD74 P04233 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27086979 1.00 NPC1 (0.38) NPC1NPSR1ALDH1A1TSHRUSP2
SCHEMBL25152612 1.00 NPC1 (0.38) NPC1NPSR1ALDH1A1TSHRUSP2
SCHEMBL27086852 0.88 NPSR1 (0.37) NPC1NPSR1ALDH1A1TSHRUSP2
SCHEMBL25152918 0.88 NPSR1 (0.37) NPC1NPSR1ALDH1A1TSHRUSP2
SCHEMBL29919584 0.88 NPSR1 (0.37) NPC1NPSR1ALDH1A1TSHRUSP2
SCHEMBL27086834 0.82 ATM (0.35) NPC1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL25152477 0.82 ATM (0.35) NPC1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL29919465 0.82 ATM (0.35) NPC1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL32686754 0.78 NPC1 (0.43) NPC1ALDH1A1MIFSIGMAR1TNIK
SCHEMBL25152956 0.76 NPC1 (0.37) NPC1ALDH1A1TSHRHPGDMIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4320105-A1 OPIOID RECEPTOR MODULATORS Epiodyne, Inc. (US) 2024-02-14 EP disclosed
CN-117425644-A Opioid receptor modulators 埃皮欧黛公司 2024-01-19 CN disclosed
WO-2022216750-A1 OPIOID RECEPTOR MODULATORS EPIODYNE, INC. (US) 2022-10-13 WO disclosed