SCHEMBL29924192

SCHEMBL29924192

CC(O)(CCl)c1ccc(Cl)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.41
CYP3A5 P20815 5/20 0.41
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CASR P41180 2/20 0.35
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
KCNH2 Q12809 1/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PDK1 Q15118 2/20 0.33
PDK2 Q15119 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251584 0.84 CYP3A4 (0.41) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL29150146 0.81 CYP3A4 (0.43) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL17186902 0.81 CYP3A4 (0.45) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL22544183 0.81 CYP3A4 (0.45) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL7943098 0.77 CYP3A4 (0.36) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL1690351 0.77 HDAC3 (0.42) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL1348538 0.76 KCNH2 (0.49) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL8805047 0.76 CYP3A4 (0.40) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL29149861 0.76 CYP3A4 (0.38) CYP3A4CYP3A5HDAC3HDAC1HDAC2
SCHEMBL24320669 0.75 CYP3A4 (0.41) CYP3A4CYP3A5HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed