SCHEMBL29925224

SCHEMBL29925224

Cn1nc(Cl)cc(Nc2ccc(C(=O)N3CCOCC3)cn2)c1=O

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
RAB9A P51151 1/20 0.56
BTK Q06187 8/20 0.51
CLK2 P49760 1/20 0.51
SRC P12931 1/20 0.49
HPGD P15428 1/20 0.48
TYK2 P29597 1/20 0.48
GRM5 P41594 5/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
LRRK2 Q5S007 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609572 1.00 KDM4E (0.56) KDM4ERAB9ABTKCLK2SRC
SCHEMBL610958 0.92 HPGD (0.57) KDM4ERAB9ABTKHPGDTYK2
SCHEMBL15906434 0.90 FASN (0.51) BTKHPGDGRM5
SCHEMBL12602961 0.90 GRM5 (0.60) KDM4ERAB9AHPGDTYK2GRM5
SCHEMBL12650334 0.89 KDM4E (0.59) KDM4ERAB9ABTKCLK2SRC
SCHEMBL608992 0.87 HPGD (0.48) KDM4ERAB9ABTKHPGDGRM5
SCHEMBL14926081 0.86 KDM4E (0.54) KDM4ERAB9ABTKCLK2SRC
SCHEMBL14926077 0.85 GRM5 (0.46) KDM4ERAB9ABTKCLK2HPGD
SCHEMBL14926064 0.85 GRM5 (0.46) KDM4ERAB9ABTKCLK2HPGD
SCHEMBL15906433 0.85 GRM5 (0.49) KDM4ERAB9ABTKHPGDGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4050012-A1 PYRIDONE BORONATES FOR THE PREPARATION OF INHIBITORS OF BTK ACTIVITY F. Hoffmann-La Roche AG (CH) 2022-08-31 EP disclosed