SCHEMBL29935989

SCHEMBL29935989

COc1c(Br)ccc2ncnc(Nc3ccc(Oc4ccn5ncnc5c4)c(C)c3)c12

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 16/20 0.64
EGFR P00533 8/20 0.60
NQO2 P16083 1/20 0.60
FECH P22830 1/20 0.60
MYH14 Q7Z406 1/20 0.60
RIPK3 Q9Y572 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27093466 1.00 ERBB2 (0.64) ERBB2EGFRNQO2FECHMYH14
SCHEMBL24167675 0.90 ERBB2 (0.64) ERBB2EGFRNQO2FECHMYH14
SCHEMBL21563124 0.89 ERBB2 (0.63) ERBB2EGFRNQO2FECHMYH14
SCHEMBL29888215 0.89 ERBB2 (0.60) ERBB2EGFRNQO2FECHMYH14
SCHEMBL29936028 0.89 ERBB2 (0.60) ERBB2EGFRNQO2FECHMYH14
SCHEMBL24167353 0.89 ERBB2 (0.60) ERBB2EGFRNQO2FECHMYH14
SCHEMBL24167673 0.86 ERBB2 (0.60) ERBB2EGFRNQO2FECHMYH14
SCHEMBL21563122 0.86 ERBB2 (0.66) ERBB2EGFRNQO2FECHMYH14
SCHEMBL26697702 0.84 ERBB2 (0.62) ERBB2EGFRNQO2FECHMYH14
SCHEMBL26006688 0.84 ERBB2 (0.63) ERBB2EGFRNQO2FECHMYH14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118459485-A Amino-substituted heterocycles for the treatment of cancers with EGFR mutations 纽威伦特公司 2024-08-09 CN disclosed
EP-4323356-A1 AMINO-SUBSTITUTED HETEROCYCLES FOR TREATING CANCERS WITH EGFR MUTATIONS Nuvalent, Inc. (US) 2024-02-21 EP disclosed
WO-2022221227-A1 AMINO-SUBSTITUTED HETEROCYCLES FOR TREATING CANCERS WITH EGFR MUTATIONS NUVALENT, INC. (US) 2022-10-20 WO disclosed