SCHEMBL29939645

SCHEMBL29939645

COc1ncc(C2CCOCC2)c2sc(NC(=O)c3ccccc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.45
ADORA2A P29274 3/20 0.45
SCD O00767 4/20 0.44
MEN1 O00255 6/20 0.43
KMT2A Q03164 6/20 0.43
ADORA3 P0DMS8 2/20 0.43
CHRM4 P08173 1/20 0.43
RXFP1 Q9HBX9 1/20 0.42
MAPT P10636 5/20 0.41
LRRK2 Q5S007 2/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
PKM P14618 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HCRTR1 O43613 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20702466 1.00 ADORA1 (0.45) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL30128173 0.89 ADORA2A (0.45) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL22027655 0.89 ADORA2A (0.45) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL22027625 0.88 ADORA2A (0.44) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL20702447 0.88 LRRK2 (0.40) ADORA1ADORA2ACHRM4MAPTLRRK2
SCHEMBL30128168 0.87 ADORA2A (0.46) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL20702422 0.87 ADORA2A (0.46) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL31256925 0.87 ADORA1 (0.44) ADORA1ADORA2ASCDMEN1KMT2A
SCHEMBL22027632 0.87 CCNE1 (0.42) ADORA1ADORA2AMEN1KMT2AMAPT
SCHEMBL30128068 0.87 CCNE1 (0.42) ADORA1ADORA2AMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997681-B Thiazolopyridine derivatives as adenosine receptor antagonists 默克专利股份公司 2022-11-15 CN disclosed