SCHEMBL29940583

SCHEMBL29940583

NC(=O)c1ccncc1-c1ccc2[nH]ccc2c1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCNC P24863 8/20 0.60
CDK8 P49336 8/20 0.60
PI4K2A Q9BTU6 2/20 0.54
IKBKB O14920 2/20 0.52
CHUK O15111 2/20 0.52
AR P10275 1/20 0.50
CYP17A1 P05093 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
BRAF P15056 1/20 0.45
CDK19 Q9BWU1 2/20 0.45
SYK P43405 1/20 0.43
PRKCQ Q04759 1/20 0.42
MAP3K11 Q16584 1/20 0.42
PIK3CD O00329 1/20 0.42
PIK3CB P42338 1/20 0.42
PIK3CG P48736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997464 0.81 PI4K2A (0.55) PI4K2AIKBKBCHUKAR
SCHEMBL28264516 0.81 PI4K2A (0.55) PI4K2AIKBKBCHUKAR
SCHEMBL29740440 0.76 AR (0.54) CCNCCDK8ARBRAFCDK19
SCHEMBL3462850 0.76 CCNC (0.56) CCNCCDK8CYP17A1CYP11B1CYP11B2
SCHEMBL30494427 0.76 CCNC (0.56) CCNCCDK8CYP17A1CYP11B1CYP11B2
SCHEMBL26463099 0.76 CCNC (0.56) CCNCCDK8CYP17A1CYP11B1CYP11B2
SCHEMBL17909801 0.75 PI4K2A (0.50) CCNCCDK8PI4K2AIKBKBCHUK
SCHEMBL31280998 0.75 CCNC (1.00) CCNCCDK8CDK19
SCHEMBL578834 0.75 AR (0.58) CCNCCDK8PI4K2AARPRKCQ
SCHEMBL28644510 0.75 CCNC (1.00) CCNCCDK8CDK19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111072634-B 1-substituted-3-substituted-5-substituted amide-1H-indole compound and preparation method and application thereof 中国医科大学 2022-07-22 CN claimed