SCHEMBL299409

SCHEMBL299409

O=C(CO)NC1CC(n2cnc3c(NCC(c4ccccc4)c4ccccc4)nc(-n4cnc(NC(=O)NCc5cccc(O)c5)c4)nc32)C(O)C1O

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.51
ADORA3 P0DMS8 8/20 0.49
ADORA1 P30542 3/20 0.38
ADORA2B P29275 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL243816 1.00 ADORA2A (0.51) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL240158 0.97 ADORA2A (0.47) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL243231 0.90 ADORA2A (0.51) ADORA2AADORA3ADORA1
SCHEMBL241855 0.89 ADORA2A (0.49) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL243007 0.89 ADORA2A (0.52) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL242018 0.88 ADORA2A (0.48) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241724 0.87 ADORA2A (0.47) ADORA2AADORA3ADORA1
SCHEMBL244368 0.86 ADORA2A (0.46) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241770 0.86 ADORA2A (0.48) ADORA2AADORA3
SCHEMBL241771 0.86 ADORA2A (0.48) ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed