SCHEMBL29948249

SCHEMBL29948249

O=c1[nH]nc2c3ccccc3[nH]c(=O)n12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HAVCR2 Q8TDQ0 2/20 0.49
HSD17B10 Q99714 1/20 0.49
KDM4E B2RXH2 4/20 0.47
CA12 O43570 2/20 0.47
CA9 Q16790 2/20 0.47
PARP1 P09874 1/20 0.47
GABRP O00591 1/20 0.47
GABRD O14764 1/20 0.47
GABRA1 P14867 1/20 0.47
GABRB1 P18505 1/20 0.47
GABRG2 P18507 1/20 0.47
GABRB3 P28472 1/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
GABRA2 P47869 1/20 0.47
GABRB2 P47870 1/20 0.47
GABRA4 P48169 1/20 0.47
GABRE P78334 1/20 0.47
GABRA6 Q16445 1/20 0.47
GABRG1 Q8N1C3 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8138057 1.00 HAVCR2 (0.49) HAVCR2HSD17B10KDM4ECA12CA9
SCHEMBL4249802 0.81 PDE3B (0.49) HSD17B10KDM4EGABRPGABRDGABRA1
SCHEMBL8137886 0.78 CHEK1 (0.56) CA12CA9ALDH1A1ADORA3LMNA
SCHEMBL8136188 0.78 FEN1 (0.51) KDM4EALDH1A1FEN1HPGDLMNA
SCHEMBL8137817 0.78 CHEK1 (0.49) HAVCR2CA12CA9CHEK1
SCHEMBL8137430 0.78 HAVCR2 (0.53) HAVCR2CA12CA9PARP1SMN1; SMN2
SCHEMBL8143260 0.78 GPR17 (0.36) HAVCR2CA12CA9PARP1GABRA1
SCHEMBL8134411 0.78 PARP1 (0.45) HAVCR2CA12CA9PARP1CHEK1
SCHEMBL8134451 0.78 FEN1 (0.51) KDM4EPARP1GABRPGABRDGABRA1
Hydrochloric Acid SCHEMBL8137045 0.76 PARP1 (0.44) HAVCR2CA12CA9PARP1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752507-B1 TRIAZOLOQUINAZOLINONE SYNTHESIS GABATHER AB (SE) 2022-11-16 EP claimed