Levomethorphan

Levomethorphan

SCHEMBL29950

COc1ccc2c(c1)[C@@]13CCCC[C@H]1[C@@H](C2)N(C)CC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GRIN2ASIGMAR1

The experimentally established mechanism targets of Levomethorphan. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2A known ✓ Q12879 8/20 1.00
SIGMAR1 known ✓ Q99720 6/20 1.00
GRIN1 Q05586 8/20 1.00
GRIN2D O15399 7/20 1.00
GRIN3B O60391 7/20 1.00
GRIN2B Q13224 7/20 1.00
GRIN2C Q14957 7/20 1.00
GRIN3A Q8TCU5 7/20 1.00
OPRM1 P35372 7/20 1.00
SLC6A4 P31645 5/20 1.00
OPRK1 P41145 4/20 1.00
TMEM97 Q5BJF2 3/20 1.00
CYP2D6 P10635 2/20 1.00
SLC6A2 P23975 2/20 1.00
SLC22A1 O15245 2/20 1.00
ADRA2A P08913 2/20 1.00
KCNH2 Q12809 2/20 1.00
MRGPRX2 Q96LB1 2/20 1.00
TSHR P16473 1/20 1.00
ADRA2C P18825 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dextromethorphan SCHEMBL29949 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL503864 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL248575 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL22722074 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL12091342 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL7380035 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL20808854 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL20809259 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL21095577 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B
Racemethorphan SCHEMBL4167360 1.00 GRIN1 (1.00) GRIN1GRIN2AGRIN2DGRIN3BGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 37833 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144765-A1 COMPOUNDS AND COMBINATIONS THEREOF FOR TREATING NEUROLOGICAL AND PSYCHIATRIC CONDITIONS ANTECIP BIOVENTURES II LLC (US) 2026-05-28 US claimed
US-20260144764-A1 COMPOUNDS AND COMBINATIONS THEREOF FOR TREATING NEUROLOGICAL AND PSYCHIATRIC CONDITIONS ANTECIP BIOVENTURES II LLC (US) 2026-05-28 US claimed
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
CN-117645615-B Method for racemizing dextromethorphan base by using ionic liquid as catalyst JIANGSU TIANHE PHARMACEUTICAL Co.,Ltd. (CN) 2026-05-26 CN claimed
CN-115927230-B Imine reductase mutant, preparation method thereof and application of imine reductase mutant in catalyzing preparation of dextromethorphan intermediate Jindawei Biotechnology (Jiangsu) Co.,Ltd. (CN) 2026-05-26 CN claimed
CN-122094687-A Compounds and combinations thereof for the treatment of neurological and psychiatric disorders 2026-05-26 CN claimed
WO-2026107265-A1 PHARMACEUTICAL DOSAGE FORMS FOR TREATING NEUROLOGICAL AND PSYCHIATRIC CONDITIONS ANTECIP BIOVENTURES II LLC (US) 2026-05-21 WO claimed
US-12629422-B2 Agave syrup formulation or suspension for active pharmaceutical agents GENEXA INC. (US) 2026-05-19 US claimed
US-20260130871-A1 COMPOUNDS AND COMBINATIONS THEREOF FOR TREATING NEUROLOGICAL AND PSYCHIATRIC CONDITIONS ANTECIP BIOVENTURES II LLC (US) 2026-05-14 US claimed
US-4446140-A Method and composition for treating mouth pain NELSON RESEARCH & DEVELOPMENT COMPANY (US) 1984-05-01 US claimed
EP-0081823-A1 Composition for reducing menstrual pain WHITBY RESEARCH, Inc. (US) 1983-06-22 EP claimed
US-4372942-A SUCROSE, CORN SYRUP, MANNITOL, GLYCERIN, SORBITOL OR SUCROSE-INVERT SUGAR MIXTURE, MOLDING BEECHAM INC. (US) 1983-02-08 US claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
US-4316888-A Method and composition of reducing pain NELSON RESEARCH & DEVELOPMENT CO. (US) 1982-02-23 US claimed
US-4260596-A Edible unit dosage form consisting of outer mannitol shell and inner liquid or gel center and method for manufacturing the same BRISTOL-MYERS COMPANY (US) 1981-04-07 US claimed
US-4221778-A ION EXCHANGE RESINS, ANTISWELLING AGENTS PENNWALT CORPORATION (US) 1980-09-09 US claimed
US-4205060-A Microcapsules containing medicament-polymer salt having a water-insoluble polymer sheath, their production and their use PENNWALT CORPORATION (US) 1980-05-27 US claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed
US-4064228-A Antigens and immunoassays for morphine and related 3-oxybenzomorphan compounds BIOLOGICAL DEVELOPMENTS, INC. (US) 1977-12-20 US claimed