SCHEMBL29953224

SCHEMBL29953224

Nc1ncc(-c2cccnc2)cc1C=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 4/20 0.57
CHEK2 O96017 1/20 0.52
FYN P06241 1/20 0.49
MKNK1 Q9BUB5 2/20 0.47
MKNK2 Q9HBH9 2/20 0.47
MEN1 O00255 1/20 0.47
PSIP1 O75475 1/20 0.47
AXL P30530 1/20 0.47
CYP2A6 P11509 5/20 0.47
CYP3A4 P08684 3/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
DYRK1A Q13627 1/20 0.44
DYRK1B Q9Y463 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
PTK2 Q05397 1/20 0.44
EGFR P00533 1/20 0.43
PDGFRB P09619 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14276837 0.83 MAP4K4 (0.49) CHEK2FYNMKNK1MKNK2AXL
SCHEMBL29955261 0.83 MAP4K4 (0.49) CHEK2FYNMKNK1MKNK2AXL
SCHEMBL18615838 0.82 MAP4K4 (0.51) CHEK2FYNMKNK1MKNK2
SCHEMBL29954696 0.82 ERN1 (0.51) ERN1CHEK2FYNEGFRPDGFRB
SCHEMBL12833995 0.81 ERN1 (0.66) ERN1CHEK2MKNK1MKNK2CYP2A6
SCHEMBL29066279 0.81 ERN1 (0.61) ERN1MKNK1MKNK2CYP2A6CYP3A4
SCHEMBL5782678 0.79 ERN1 (0.61) ERN1MKNK1MKNK2CYP2A6CYP3A4
SCHEMBL712179 0.78 FYN (0.58) CHEK2FYNMKNK1MKNK2MEN1
SCHEMBL2556015 0.78 CHEK2 (0.52) CHEK2FYNMEN1PDGFRBPDGFRA
SCHEMBL16835804 0.76 FYN (0.52) ERN1CHEK2FYNMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed