SCHEMBL29954034

SCHEMBL29954034

COc1cccc2cc(B(O)O)n(C(=O)OC(C)(C)C)c12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.41
NR1H2 P55055 11/20 0.39
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
CCR2 P41597 1/20 0.35
NR1H3 Q13133 3/20 0.35
TGFBR1 P36897 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
LMNA P02545 1/20 0.34
RECQL P46063 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13280504 1.00 BACE1 (0.41) BACE1NR1H2CA12CA9CCR2
SCHEMBL13515301 0.85 NR1H2 (0.40) NR1H2CA12CA9NR1H3TGFBR1
SCHEMBL2873473 0.84 NR1H2 (0.40) NR1H2CA12CA9NR1H3
SCHEMBL4242068 0.84 NR1H2 (0.40) BACE1NR1H2CA12CA9CCR2
SCHEMBL15431762 0.83 BACE1 (0.43) BACE1NR1H2CA12CA9CCR2
SCHEMBL759123 0.83 NR1H2 (0.40) BACE1NR1H2CA12CA9NR1H3
SCHEMBL30016078 0.83 NR1H2 (0.40) BACE1NR1H2CA12CA9NR1H3
SCHEMBL18567358 0.82 BACE1 (0.44) BACE1NR1H2CA12CA9CCR2
SCHEMBL2926879 0.80 NR1H2 (0.40) NR1H2CA12CA9CCR2NR1H3
SCHEMBL1550715 0.78 PDE4B (0.34) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4168002-A1 METHODS FOR DELAYING, PREVENTING, AND TREATING ACQUIRED RESISTANCE TO RAS INHIBITORS Revolution Medicines, Inc. (US) 2023-04-26 EP disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed