SCHEMBL29955085

SCHEMBL29955085

Cc1ccc2c(C=O)n[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 6/20 0.46
CHEK1 O14757 5/20 0.43
CDK1 P06493 1/20 0.43
CDK4 P11802 1/20 0.43
CCNA2 P20248 1/20 0.43
CCND1 P24385 1/20 0.43
CDK2 P24941 1/20 0.43
CCND3 P30281 1/20 0.43
MAP2K7 O14733 1/20 0.41
PIM3 Q86V86 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
TTK P33981 1/20 0.38
MAPK1 P28482 2/20 0.38
MAP2K4 P45985 2/20 0.38
MAPKAPK3 Q16644 2/20 0.38
MAPK6 Q16659 2/20 0.38
MAPKAPK2 P49137 1/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
KIF11 P52732 1/20 0.38
KDR P35968 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15304355 1.00 ITK (0.46) ITKCHEK1CDK1CDK4CCNA2
SCHEMBL5953047 0.86 MAP2K4 (0.49) ITKCHEK1MAPK1MAP2K4MAPKAPK3
SCHEMBL3538242 0.80 TTK (0.54) CHEK1CDK1CDK4CCNA2CCND1
SCHEMBL13632256 0.79 GRIA1 (0.36) CHEK1CDK1CDK4CCNA2CCND1
SCHEMBL27384927 0.79 PARP1 (0.42) CHEK1PARP1PIM1RPS6KA3
SCHEMBL29497531 0.79 PDPK1 (0.58) CHEK1CDK2PIM3KDRPIM1
SCHEMBL29956078 0.79 AXL (0.45) CHEK1KDRPARP1
SCHEMBL3537177 0.79 MAP2K4 (0.51) ITKCHEK1CDK1CDK4CCNA2
SCHEMBL29935743 0.79 MAP2K4 (0.51) ITKCHEK1CDK1CDK4CCNA2
SCHEMBL29955404 0.79 PDPK1 (0.54) CHEK1CDK4CCND1CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed