SCHEMBL29960435

SCHEMBL29960435

O=C(NC1CC(O)C1)c1ccc(N2CCNCC2)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 4/20 0.49
MAPT P10636 5/20 0.47
ALDH1A1 P00352 3/20 0.47
POLB P06746 2/20 0.43
PARP1 P09874 1/20 0.42
TNK2 Q07912 1/20 0.42
TNK1 Q13470 1/20 0.42
BMPR1B O00238 1/20 0.41
BMPR1A P36894 1/20 0.41
TGFBR1 P36897 1/20 0.41
ACVRL1 P37023 1/20 0.41
ACVR1 Q04771 1/20 0.41
GAA P10253 1/20 0.41
MAPKAPK2 P49137 1/20 0.41
HPGD P15428 2/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.40
HPGDS O60760 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29115574 1.00 USP30 (0.49) USP30MAPTALDH1A1POLBPARP1
SCHEMBL29115395 1.00 USP30 (0.49) USP30MAPTALDH1A1POLBPARP1
SCHEMBL29115394 1.00 USP30 (0.49) USP30MAPTALDH1A1POLBPARP1
SCHEMBL531747 0.89 USP30 (0.54) USP30MAPTALDH1A1POLBPARP1
Hydrochloric Acid SCHEMBL709154 0.88 USP30 (0.53) USP30MAPTALDH1A1POLBPARP1
SCHEMBL29085179 0.82 USP30 (0.56) USP30MAPTALDH1A1POLBHPGD
SCHEMBL29085200 0.82 USP30 (0.56) USP30MAPTALDH1A1POLBHPGD
SCHEMBL29960478 0.82 USP30 (0.56) USP30MAPTALDH1A1POLBHPGD
SCHEMBL29085175 0.82 USP30 (0.56) USP30MAPTALDH1A1POLBHPGD
SCHEMBL531792 0.80 MAPT (0.50) MAPTALDH1A1PARP1TNK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116710433-A Selective PARP1 inhibitor and application thereof 成都百裕制药股份有限公司 2023-09-05 CN disclosed
WO-2022222966-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2022-10-27 WO disclosed