SCHEMBL29967102

SCHEMBL29967102

COc1ccc(Cl)c(Cl)c1[C@H]1C[C@@H](C(O)CCO)N(C(=O)O)C1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.41
HTR2C P28335 9/20 0.41
HTR2B P41595 7/20 0.41
KDM4E B2RXH2 3/20 0.33
DRD2 P14416 1/20 0.32
ALDH1A1 P00352 2/20 0.31
TNF P01375 1/20 0.30
RORC P51449 1/20 0.30
CYP2D6 P10635 1/20 0.30
MTNR1B P49286 1/20 0.30
S1PR1 P21453 1/20 0.30
S1PR5 Q9H228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217133 1.00 HTR2A (0.41) HTR2AHTR2CHTR2BKDM4EDRD2
SCHEMBL23217394 0.93 HTR2A (0.42) HTR2AHTR2CHTR2BKDM4EDRD2
SCHEMBL23227412 0.87 HTR2A (0.40) HTR2AHTR2CHTR2B
SCHEMBL23217435 0.83 HTR2C (0.45) HTR2AHTR2CHTR2BKDM4EDRD2
SCHEMBL23217052 0.83 HTR2A (0.39) HTR2AHTR2CHTR2BDRD2
SCHEMBL23217368 0.83 HTR2A (0.36) HTR2AHTR2CHTR2BCYP2D6MTNR1B
SCHEMBL23217075 0.80 HTR2A (0.47) HTR2AHTR2CHTR2BKDM4EDRD2
SCHEMBL23227255 0.80 HTR2A (0.41) HTR2AHTR2CHTR2B
SCHEMBL23217149 0.79 HTR2C (0.45) HTR2AHTR2CHTR2BKDM4EDRD2
SCHEMBL23217480 0.78 HTR2C (0.44) HTR2AHTR2CHTR2BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114828963-A Arylheterobicyclic compounds as Kv1.3 potassium SHAKER channel blockers D·E·萧尔研究有限责任公司 2022-07-29 CN disclosed