SCHEMBL29970478

SCHEMBL29970478

Nc1nc2ccc(-c3nc(N4CCOCC4)nc(N4CCOCC4)n3)cc2s1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 17/20 1.00
NPC1 O15118 2/20 0.64
MAPT P10636 2/20 0.64
RAB9A P51151 2/20 0.64
SMN1; SMN2 Q16637 2/20 0.64
TP53 P04637 1/20 0.64
ALOX15 P16050 1/20 0.64
PIK3R1 P27986 3/20 0.59
MTOR P42345 3/20 0.59
PIK3CD O00329 3/20 0.58
PIK3CG P48736 3/20 0.58
PIK3CB P42338 2/20 0.58
PI4KA P42356 3/20 0.52
PI4KB Q9UBF8 3/20 0.52
PIP5K1C O60331 1/20 0.52
GAA P10253 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28617302 1.00 PIK3CA (1.00) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL29970161 0.91 PIK3CA (0.83) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL28600969 0.89 PIK3CA (1.00) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL29971056 0.89 PIK3CA (0.84) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL30012232 0.89 PIK3CA (1.00) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL30011161 0.89 PIK3CA (1.00) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL28614234 0.89 PIK3CA (0.78) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL30012022 0.89 PIK3CA (0.78) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL28602635 0.89 PIK3CA (1.00) PIK3CANPC1MAPTRAB9ASMN1; SMN2
SCHEMBL25259671 0.83 NPC1 (0.82) PIK3CANPC1MAPTRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200969-B PI3K alpha selective inhibitor and preparation method and application thereof 中国药科大学 2022-11-25 CN disclosed
WO-2022242321-A1 PI3Kα SELECTIVE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 中国药科大学 2022-11-24 WO disclosed