SCHEMBL29975585

SCHEMBL29975585

CC(C)(C)OC(=O)Nc1ccnc(C(C)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 1/20 0.50
SMARCA4 P51532 1/20 0.50
CYP17A1 P05093 3/20 0.44
PRKCI P41743 1/20 0.44
ATR Q13535 1/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
NAMPT P43490 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAP4K4 O95819 1/20 0.42
SYK P43405 1/20 0.42
RAF1 P04049 2/20 0.41
BRAF P15056 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
SREBF2 Q12772 1/20 0.40
RORC P51449 1/20 0.40
MAPK14 Q16539 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16121247 1.00 SMARCA2 (0.50) SMARCA2SMARCA4CYP17A1PRKCIATR
SCHEMBL21614653 0.91 SMARCA2 (0.60) SMARCA2SMARCA4CYP17A1PRKCIATR
SCHEMBL29099947 0.84 MAP4K4 (0.44) SMARCA2SMARCA4CYP17A1PRKCIATR
SCHEMBL28400383 0.83 ATR (0.45) SMARCA2SMARCA4CYP17A1PRKCIATR
SCHEMBL16369790 0.82 SMARCA2 (0.51) SMARCA2SMARCA4PRKCIRAF1BRAF
SCHEMBL16055308 0.81 SMARCA2 (0.57) SMARCA2SMARCA4CYP17A1ATRCA12
SCHEMBL1501665 0.81 SMARCA2 (0.57) SMARCA2SMARCA4CYP17A1ATRCA12
SCHEMBL30293080 0.81 SMARCA2 (0.57) SMARCA2SMARCA4CYP17A1ATRCA12
SCHEMBL2596875 0.79 AR (0.56) SMARCA2SMARCA4CYP17A1ATRCA12
SCHEMBL29383469 0.79 AR (0.56) SMARCA2SMARCA4CYP17A1ATRCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12433895-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2025-10-07 US disclosed
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE PHARMARESROUCES (SHANGHAI) CO., LTD. (CN) 2024-10-10 US disclosed
US-11844758-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2023-12-19 US disclosed
CN-117120427-A MALT1 inhibitor and preparation method and application thereof 上海拓界生物医药科技有限公司 2023-11-24 CN disclosed
US-20220354856-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE SERVIER PHARMACEUTICALS LLC 2022-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12433895-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT SMARCA2 1910/4885SMARCA4 2048/4885CYP17A1 2927/4885
US-11844758-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT SMARCA2 1910/4885SMARCA4 2048/4885CYP17A1 2927/4885
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT SMARCA2 1910/4885SMARCA4 2048/4885CYP17A1 2927/4885
US-20220354856-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT SMARCA2 1910/4885SMARCA4 2048/4885CYP17A1 2927/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.