SCHEMBL29975823

SCHEMBL29975823

Cc1c(N)ccc2c1OC(F)(F)O2

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.44
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
PIK3CA P42336 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14007746 1.00 ADORA2A (0.44) ADORA2ACYP3A4TSHRPIK3CA
SCHEMBL12744378 0.83 ADORA2A (0.38) ADORA2A
Hydrochloric Acid SCHEMBL10371157 0.83 ADORA2A (0.39) ADORA2A
SCHEMBL21901486 0.82 ADORA2A (0.38) ADORA2A
SCHEMBL21603470 0.80 ADORA2A (0.43) ADORA2A
SCHEMBL21532908 0.80 ESR1 (0.42) ADORA2A
SCHEMBL13395585 0.80 ADORA2A (0.38) ADORA2A
SCHEMBL12879229 0.80 ADORA2A (0.37) ADORA2A
SCHEMBL3055306 0.80 ADORA2A (0.37) ADORA2A
SCHEMBL23461927 0.77 ADORA2A (0.35) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069216-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF CYSTIC FIBROSIS Flatley Discovery Lab, LLC (US) 2022-10-12 EP disclosed