SCHEMBL29978161

SCHEMBL29978161

CC(C)(C)OC(=O)N1CCc2sc(C(N)=NO)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.50
HDAC6 Q9UBN7 4/20 0.49
ESR2 Q92731 1/20 0.48
ADORA1 P30542 2/20 0.45
BRD4 O60885 1/20 0.44
CREBBP Q92793 1/20 0.44
MAPT P10636 3/20 0.41
KDM4E B2RXH2 1/20 0.41
F2 P00734 1/20 0.41
TPSAB1 Q15661 1/20 0.41
TPSD1 Q9BZJ3 1/20 0.41
TPSG1 Q9NRR2 1/20 0.41
MAPK1 P28482 1/20 0.40
NAMPT P43490 1/20 0.37
NPC1 O15118 1/20 0.36
PLA2G1B P04054 1/20 0.36
RAB9A P51151 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
GRAMD1A Q96CP6 1/20 0.36
MKNK1 Q9BUB5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978014 0.91 NR1H2 (0.50) NR1H2HDAC6ESR2ADORA1MAPT
SCHEMBL6421478 0.88 NR1H2 (0.54) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL743782 0.84 HDAC6 (0.54) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL8555269 0.84 HDAC6 (0.54) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL978284 0.83 HDAC6 (0.59) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL8558892 0.83 NR1H2 (0.51) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL1174513 0.82 HDAC6 (0.72) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL6422061 0.81 NR1H2 (0.52) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL14876121 0.81 NR1H2 (0.60) NR1H2HDAC6ESR2ADORA1BRD4
SCHEMBL1174301 0.81 ADORA1 (0.57) NR1H2HDAC6ESR2ADORA1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed