SCHEMBL29978217

SCHEMBL29978217

O=C(NCc1ccc(F)cc1)N1CCc2sc(-c3noc(C(F)(F)F)n3)cc2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
NPC1 O15118 1/20 0.50
HDAC6 Q9UBN7 14/20 0.45
HDAC1 Q13547 8/20 0.45
HDAC8 Q9BY41 6/20 0.45
HDAC5 Q9UQL6 2/20 0.43
HDAC4 P56524 6/20 0.43
MAPK1 P28482 1/20 0.43
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42
TUBA4A P68366 1/20 0.42
TUBB4B P68371 1/20 0.42
TUBB3 Q13509 1/20 0.42
TUBB2A Q13885 1/20 0.42
TUBB8 Q3ZCM7 1/20 0.42
TUBA3E Q6PEY2 1/20 0.42
TUBA1A Q71U36 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978199 0.93 KMT2A (0.50) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29978595 0.92 HDAC6 (0.50) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29978276 0.91 MAPK1 (0.46) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29978083 0.88 NPC1 (0.47) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29978027 0.88 HDAC6 (0.53) HDAC6HDAC1HDAC8HDAC4MAPK1
SCHEMBL29978607 0.87 HDAC6 (0.43) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29978106 0.86 KMT2A (0.50) KMT2AMEN1NPC1HDAC6HDAC1
SCHEMBL29977967 0.86 HDAC4 (0.50) HDAC6HDAC1HDAC8HDAC4HDAC2
SCHEMBL29977874 0.86 HDAC4 (0.45) HDAC6HDAC1HDAC8HDAC5HDAC4
SCHEMBL29978188 0.86 HDAC4 (0.41) HDAC6HDAC1HDAC8HDAC5HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed