SCHEMBL29987607

SCHEMBL29987607

COc1cccc(-c2cncc(C=O)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 5/20 0.49
CYP11B2 P19099 5/20 0.49
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2C9 P11712 3/20 0.49
ERN1 O75460 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A1 P04798 2/20 0.46
CYP1B1 Q16678 2/20 0.46
PDGFRB P09619 1/20 0.46
PDGFRA P16234 1/20 0.46
DAPK3 O43293 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
DYRK1A Q13627 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
KDR P35968 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16180188 1.00 CYP11B1 (0.49) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL16180062 0.88 CYP11B1 (0.53) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL2591901 0.84 ERN1 (0.55) CYP1A2CYP3A4CYP2C9ERN1ALDH1A1
SCHEMBL12108683 0.84 CYP11B1 (0.65) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL2318682 0.83 MAP4K4 (0.55) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL28881249 0.81 CYP11B1 (0.46) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL29597243 0.81 CYP11B1 (0.50) CYP11B1CYP11B2DYRK1A
SCHEMBL29066294 0.81 CYP11B1 (0.50) CYP11B1CYP11B2DYRK1A
SCHEMBL29987430 0.81 CYP11B1 (0.46) CYP11B1CYP11B2CYP1A2CYP3A4CYP2C9
SCHEMBL2581063 0.79 DRD1 (0.64) CYP1A2CYP3A4CYP2C9ERN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304591-B Bridged ring steroid synthetase inhibitor and preparation method and application thereof 广州中医药大学(广州中医药研究院) 2024-10-01 CN disclosed
CN-115304591-A Bridged steroid synthetase inhibitor and preparation method and application thereof 广州中医药大学(广州中医药研究院) 2022-11-08 CN disclosed