SCHEMBL299893

SCHEMBL299893

CN1C(=O)CSc2cc(-c3ccc(CC(C#N)NC(=O)C4(NC(=O)O)CCOCC4)cc3)ccc21.CN1C(=O)CSc2cc(-c3ccc(CC(NC(=O)C4(NC(=O)O)CCOCC4C(C)(C)C)C(N)=O)cc3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSC P53634 20/20 0.46
CTSK P43235 4/20 0.40
KCNH2 Q12809 1/20 0.36
LTB4R Q15722 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299129 0.89 CTSC (0.49) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL299257 0.86 CTSC (0.56) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL299829 0.86 CTSC (0.42) CTSCCTSK
SCHEMBL9886054 0.80 CTSC (0.52) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL9886053 0.79 CTSC (0.40) CTSCCTSK
SCHEMBL2885836 0.77 CTSC (0.72) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2885832 0.77 CTSC (0.72) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL298828 0.75 CTSC (0.61) CTSCCTSKKCNH2LTB4RLTB4R2
SCHEMBL2885772 0.75 CTSC (0.47) CTSCCTSK
SCHEMBL2888765 0.73 CTSC (0.78) CTSCCTSKKCNH2LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed