SCHEMBL29989352

SCHEMBL29989352

Cc1nc(N(C)c2ccc3c(c2)cc(C)n3C)c2ccccc2n1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.57
PDGFRB P09619 3/20 0.57
KDR P35968 3/20 0.57
HDAC1 Q13547 8/20 0.45
HDAC8 Q9BY41 7/20 0.45
HDAC6 Q9UBN7 7/20 0.45
PDE5A O76074 2/20 0.45
HDAC11 Q96DB2 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29988823 0.88 EGFR (0.55) EGFRPDGFRBKDRPDE5AABCG2
SCHEMBL28491414 0.88 EGFR (0.55) EGFRPDGFRBKDRPDE5AABCG2
SCHEMBL23037568 0.84 EGFR (0.56) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL30367299 0.81 CYP1A2 (0.40) EGFRPDGFRBKDRCYP1A2
SCHEMBL2256659 0.80 EGFR (0.54) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL3115859 0.76 EGFR (0.74) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL19789164 0.76 EGFR (0.74) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL19789183 0.75 EGFR (0.62) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL2259608 0.73 EGFR (0.74) EGFRPDGFRBKDRHDAC1HDAC8
SCHEMBL2256177 0.73 EGFR (0.70) EGFRPDGFRBKDRHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115417860-B Quinazoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2023-10-20 CN disclosed
CN-111892581-B Quinazoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2022-12-27 CN disclosed
CN-115417860-A Quinazoline derivative with anti-tumor activity and synthesis method and application thereof 中国药科大学 2022-12-02 CN disclosed