SCHEMBL299901

SCHEMBL299901

NC(=O)C(=O)[C@@H](Cc1ccccc1)NC(=O)C1CCC(=O)N1Cc1cc(F)cc(F)c1

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 10/20 0.74
ITGB1 P05556 9/20 0.56
ITGA4 P13612 9/20 0.56
P2RX7 Q99572 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289632 1.00 CAPN1 (0.74) CAPN1ITGB1ITGA4P2RX7
SCHEMBL288113 1.00 CAPN1 (0.74) CAPN1ITGB1ITGA4P2RX7
SCHEMBL1612415 1.00 CAPN1 (0.74) CAPN1ITGB1ITGA4P2RX7
SCHEMBL1612618 0.93 CAPN1 (0.72) CAPN1ITGB1ITGA4P2RX7
SCHEMBL1612831 0.93 CAPN1 (0.72) CAPN1ITGB1ITGA4P2RX7
SCHEMBL1613552 0.93 CAPN1 (0.72) CAPN1ITGB1ITGA4P2RX7
SCHEMBL1612818 0.91 CAPN1 (0.78) CAPN1ITGB1ITGA4P2RX7
SCHEMBL289988 0.91 CAPN1 (0.78) CAPN1ITGB1ITGA4P2RX7
SCHEMBL289223 0.91 CAPN1 (0.78) CAPN1ITGB1ITGA4P2RX7
SCHEMBL288910 0.91 CAPN1 (0.88) CAPN1ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427429-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS Abbott GmbH & Co. KG (DE) 2012-03-14 EP disclosed
WO-2010128102-A1 CARBOXAMIDE COMPOUNDS AND THEIR USE AS CALPAIN INHIBITORS ABBOTT GMBH & CO. KG (DE) 2010-11-11 WO disclosed