SCHEMBL299918

SCHEMBL299918

CCCS(=O)(=O)c1ccc(-c2ccc(C[C@@H](C#N)NC(=O)C3(NC(=O)OC(C)(C)C)CCOCC3)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSC P53634 16/20 0.48
KCNH2 Q12809 2/20 0.47
LTB4R Q15722 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.47
CTSK P43235 4/20 0.41
LGMN Q99538 1/20 0.40
CTSS P25774 1/20 0.38
RET P07949 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSF Q9UBX1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2890537 0.94 CTSC (0.50) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2890536 0.94 CTSC (0.50) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2893243 0.89 CTSC (0.49) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2893241 0.89 CTSC (0.49) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2891122 0.87 CTSC (0.51) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2891123 0.87 CTSC (0.51) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL7873696 0.86 CTSC (0.47) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL16485747 0.86 CTSC (0.49) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL7864104 0.86 CTSC (0.52) CTSCKCNH2LTB4RLTB4R2CTSK
SCHEMBL2890491 0.86 CTSC (0.52) CTSCKCNH2LTB4RLTB4R2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427445-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 AstraZeneca AB (SE) 2012-03-14 EP disclosed
WO-2010128324-A1 SUBSTITUTED 1-CYANOETHYLHETEROCYCLYLCARBOXAMIDE COMPOUNDS 750 ASTRAZENECA AB (SE) 2010-11-11 WO disclosed