Pyridarone

Pyridarone

SCHEMBL29993452

c1ccc2oc(-c3ccncc3)cc2c1

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.62
ADRA2A P08913 2/20 0.56
MAOA P21397 3/20 0.54
ALOX5 P09917 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA9 Q16790 1/20 0.54
NPC1 O15118 4/20 0.53
RAB9A P51151 3/20 0.53
MAPT P10636 1/20 0.53
ADORA2A P29274 1/20 0.51
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 2/20 0.50
CYP19A1 P11511 1/20 0.50
GRM4 Q14833 1/20 0.50
CYP2D6 P10635 1/20 0.50
HPGD P15428 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridarone SCHEMBL2109298 1.00 MAOB (0.62) MAOBADRA2AMAOAALOX5CA1
Pyridine SCHEMBL28895931 0.89 MAOB (0.59) MAOBADRA2AMAOAALOX5CA1
SCHEMBL4659168 0.84 MAOB (0.78) MAOBADRA2AMAOAALOX5CA1
SCHEMBL31105656 0.84 MAOB (0.71) MAOBADRA2AMAOAALOX5CA1
SCHEMBL731363 0.84 MAOB (0.71) MAOBADRA2AMAOAALOX5CA1
SCHEMBL7125605 0.81 MAOB (0.68) MAOBADRA2AMAOAALOX5CA1
SCHEMBL3075181 0.81 ADORA2A (0.55) MAOBADRA2AMAOAALOX5CA1
SCHEMBL15446906 0.81 MAOB (0.47) MAOBADRA2AMAOAALOX5CA1
SCHEMBL2960606 0.80 MAOB (0.54) MAOBADRA2AMAOAALOX5CA1
SCHEMBL29993564 0.80 MAOB (0.54) MAOBADRA2AMAOAALOX5CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115160310-B Alternanthene derivatives as CDK2/Topo I inhibitors, preparation method thereof and antitumor application thereof 中国人民解放军北部战区总医院 2023-06-23 CN disclosed
CN-115160310-A Sinomenine derivatives as CDK2/Topo I inhibitor, and preparation method and anti-tumor application thereof 中国人民解放军北部战区总医院 2022-10-11 CN disclosed