SCHEMBL30002640

SCHEMBL30002640

COC(=O)c1cccc2ccc(C)nc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.66
KDM4E B2RXH2 4/20 0.62
MAPT P10636 2/20 0.52
GAA P10253 2/20 0.52
METAP2 P50579 1/20 0.51
CD38 P28907 1/20 0.50
ALDH1A1 P00352 1/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TP53 P04637 1/20 0.49
KMT2A Q03164 1/20 0.48
ATM Q13315 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
GLO1 Q04760 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13740437 1.00 PARP1 (0.66) PARP1KDM4EMAPTGAAMETAP2
SCHEMBL31429914 0.83 KDM4E (0.48) PARP1KDM4EMAPTGAAALDH1A1
SCHEMBL4631555 0.82 MCHR1 (0.54) PARP1KDM4EGAAALDH1A1LMNA
SCHEMBL12768665 0.82 KDM4E (0.47) PARP1KDM4EGAAALDH1A1LMNA
SCHEMBL27772010 0.81 PARP1 (0.72) PARP1KDM4EMAPTGAAMETAP2
SCHEMBL5319765 0.81 PARP1 (0.72) PARP1KDM4EMAPTGAAMETAP2
SCHEMBL29412561 0.81 PARP1 (0.72) PARP1KDM4EMAPTGAAMETAP2
SCHEMBL10566270 0.80 KDM4E (0.49) PARP1KDM4EMAPTGAAMETAP2
SCHEMBL422282 0.79 PARP1 (1.00) PARP1MAPTGAAMETAP2CD38
SCHEMBL21816896 0.79 PARP1 (0.70) PARP1KDM4EMAPTGAAMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed